๐ The adamantane-derived bananins are potent inhibitors of the helicase activities and replication of SARS coronavirus
Bananins are a class of antiviral compounds with a unique structural signature incorporating a trioxa-adamantane moiety covalently bound to a pyridoxal derivative. Six members of this class of compounds: bananin, iodobananin, vanillinbananin, ansabananin, eubananin, and adeninobananin were synthesized and tested as inhibitors of the SARS Coronavirus (SCV) helicase. Bananin, iodobananin, vanillinbananin, and eubananin were effective inhibitors of the ATPase activity of the SCV helicase with IC50 values in the range 0.5-3 ฮผM. A similar trend, though at slightly higher inhibitor concentrations, was observed for inhibition of the helicase activities, using a FRET-based fluorescent assay. In a cell culture system of SCV, bananin exhibited an EC50 of less than 10 ฮผM and a CC50 of over 300 ฮผM. Kinetics of inhibition are consistent with bananin inhibiting an intracellular process or processes involved in SCV replication. ยฉ 2005 Elsevier Ltd
keywords
๐ cell culture (240)
author
๐ค Tanner, Julian A.
๐ค Zheng, Bo Jian
๐ค Zhou, Jie
๐ค Watt, Rory M.
๐ค Jiang, Jie Qing
๐ค Wong, Kin Ling
๐ค Lin, Yong Ping
๐ค Lu, Lin Yu
๐ค He, Ming Liang
๐ค Kung, Hsiang Fu
๐ค Kesel, Andreas J.
๐ค Huang, Jian Dong
year
โฐ 2005
journal
๐ Chemistry and Biology
issn
๐ 10745521
volume
12
number
3
page
303-311
citedbycount
63
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